A Menin-MLL Inhibitor Induces Specific Chromatin Changes and Eradicates Disease in Models of MLL-Rearranged Leukemia - ScienceDirect
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Inhibition of the Menin (MEN1) and MLL (MLL1, KMT2A) interaction is a potential therapeutic strategy for MLL-rearranged (MLL-r) leukemia. Structure-ba…
A Menin-MLL Inhibitor Induces Specific Chromatin Changes and
A Menin-MLL Inhibitor Induces Specific Chromatin Changes and
Designed to kill: novel menin-MLL inhibitors target MLL-rearranged
Biochemical perspectives on targeting KMT2 methyltransferases in
Frontiers Rewiring the Epigenetic Networks in MLL-Rearranged
Dissection of the MEF2D-IRF8 transcriptional circuit dependency in
High-Affinity Small-Molecule Inhibitors of the Menin-Mixed Lineage
Complementary activities of DOT1L and Menin inhibitors in MLL
Paralog-specific signaling by IRAK1/4 maintains MyD88-independent
MLL::AF9 degradation induces rapid changes in transcriptional
A Menin-MLL Inhibitor Induces Specific Chromatin Changes and
Recent Progress of Small Molecule Menin–MLL Interaction Inhibitors
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